Research Topic

high-throughput

7 publications exploring this topic

2025

2025
cited5

AIMNet2-rxn: A Machine Learned Potential for Generalized Reaction Modeling on a Millions-of-Pathways Scale

Anstine D. M., Zhao Q., Zubatiuk R., Zhang S., Singla V., Nikitin F., Savoie B. M., Isayev O.

(2025)

Reactions Reactivity
Ml Potentials
Quantum Chemistry

AIMNet2-rxn is a machine-learned interatomic potential trained on 4.7 10^6 range-separated DFT calculations that accelerates reaction modeling by about six orders of magnitude while retaining approximately 1–2 kcal/mol accuracy along reaction coordinates. By leveraging three‑dimensional chemical information and a batched nudged elastic band (BNEB) method, the model searches millions of reaction pathways and enables high‑throughput mechanistic analysis for complex transformations such as glucose pyrolysis.

DOI
2025
cited3

Transferable Machine Learning Interatomic Potential for Pd-Catalyzed Cross-Coupling Reactions

Anstine D., Zubatyuk R., Gallegos L., Paton R., Wiest O., Nebgen B., Jones T., Gomes G., Tretiak S., Isayev O.

(2025)

Ml Potentials
Reactions Reactivity
Experiment Automation
Materials Informatics

Finding efficient substrate-catalyst combinations for palladium-catalyzed cross-coupling reactions remains a critical challenge in synthetic chemistry, with broad implications for pharmaceutical and materials manufacturing.

DOI
2025

High-throughput electronic property prediction of cyclic molecules with 3D-enhanced machine learning

Zheng P., Isayev O.

Chemical Science, 16, 20553–20563 (2025)

Ring Vault contains 201 546 cyclic molecules across 11 elements.

DOI

2024

2024
cited1

In silico screening of LRRK2 WDR domain inhibitors using deep docking and free energy simulations

Gutkin E., Gusev F., Gentile F., Ban F., Koby S. B., Narangoda C., Isayev O., Cherkasov A., Kurnikova M. G.

(2024)

Drug Discovery
Experiment Automation

The Critical Assessment of Computational Hit-Finding Experiments (CACHE) Challenge series is focused on identifying small molecule inhibitors of protein targets using computational methods.

DOI
2024
cited85

Exploring the frontiers of condensed-phase chemistry with a general reactive machine learning potential

Zhang S., Makoś M. Z., Jadrich R. B., Kraka E., Barros K., Nebgen B. T., Tretiak S., Isayev O., Lubbers N., Messerly R. A., Smith J. S.

Nature Chemistry, 16, 727–734 (2024)

Ml Potentials
Experiment Automation

Abstract Atomistic simulation has a broad range of applications from drug design to materials discovery.

DOI

2023

2023

In silico screening of LRRK2 WDR domain inhibitors using deep docking and free energy simulations

Gutkin E., Gusev F., Gentile F., Ban F., Koby S. B., Narangoda C., Isayev O., Cherkasov A., Kurnikova M. G.

(2023)

Drug Discovery
Experiment Automation

The Critical Assessment of Computational Hit-Finding Experiments (CACHE) Challenge is focused on identifying small molecule inhibitors of protein targets using computational methods.

DOI
2023

The Challenge of Balancing Model Sensitivity and Robustness in Predicting Yields: A Benchmarking Study of Amide Coupling Reactions

Liu Z., Moroz Y. S., Isayev O.

(2023)

Reactions Reactivity
Experiment Automation

Accurate prediction of reaction yield is the holy grail for computer-assisted synthesis, but current models have failed to generalize to large literature datasets.

DOI